Kun Sándor
DE >
TTKAssistant professor 2018-
Name: Kun Sándor
Degree
- PhD, Debreceni Egyetem (2014)
Publication list
2023
Kun, S.,
Mathomes, R.,
Docsa, T.,
Somsák, L.,
Hayes, J.:
Design and Synthesis of 3-(β-D-Glucopyranosyl)-4-amino/4-guanidino Pyrazole Derivatives and Analysis of Their Glycogen Phosphorylase Inhibitory Potential.
Molecules. 28 (7), 1-19, 2023.
Journal metrics:
Q1 Analytical Chemistry
Q1 Chemistry (miscellaneous)
Q2 Drug Discovery
Q2 Medicine (miscellaneous)
Q3 Molecular Medicine
Q2 Organic Chemistry
Q1 Pharmaceutical Science
Q2 Physical and Theoretical Chemistry
2022
2021
Sipos, Á.,
Szennyes, E.,
Hajnal, É.,
Kun, S.,
Szabó, E.,
Uray, K.,
Somsák, L.,
Docsa, T.,
Bokor, É.:
Dual-Target Compounds against Type 2 Diabetes Mellitus: proof of Concept for Sodium Dependent Glucose Transporter (SGLT) and Glycogen Phosphorylase (GP) Inhibitors.
Pharmaceuticals. 14 (4), 1-27, 2021.
Journal metrics:
Q1 Drug Discovery
Q2 Molecular Medicine
Q1 Pharmaceutical Science
Tsagkarakou, A.,
Chasapi, S.,
Koulas, S.,
Tsialtas, I.,
Kyriakis, E.,
Drakou, C.,
Kun, S.,
Somsák, L.,
Spyroulias, G.,
Psarra, A.,
Leonidas, D.:
Structure activity relationship of the binding of p-coumaroyl glucose to glycogen phosphorylase and its effect on hepatic cell metabolic pathways.
European Journal of Medicinal Chemistry Reports. 3 1-11, 2021.
2020
Gorliczay, E.,
Tamás, J.,
Kun, S.,
Huzsvai, L.,
Bárány, L.:
Examination and statistical evaluation of physico-chemical parameters of windrow composting.
Agrártud. Közl. 1 33-38, 2020.
Kiss, N.,
Nagy, P.,
Tóth, F.,
Gorliczay, E.,
Madar, L.,
Kun, S.,
Tamás, J.:
Improving the water management properties of different soil type.
In: A klímaváltozás kihívásai a következő évtizedekben : előadások kivonatai, Szent István Egyetem, Keszthely, 54, 2020.
Kyriakis, E.,
Karra, A.,
Papaioannou, O.,
Solovou, T.,
Skamnaki, V.,
Liggri, P.,
Zographos, S.,
Szennyes, E.,
Bokor, É.,
Kun, S.,
Psarra, A.,
Somsák, L.,
Leonidas, D.:
The architecture of hydrogen and sulfur α-hole interactions explain differences in the inhibitory potency of C-β-d-glucopyranosyl thiazoles, imidazoles and an N-β-d glucopyranosyl tetrazole for human liver glycogen phosphorylase and offer new insights to structure-based design.
Bioorg. Med. Chem. 28 (1), 1-10, 2020.
Journal metrics:
Q3 Biochemistry
Q2 Clinical Biochemistry
Q2 Drug Discovery
Q3 Molecular Biology
Q3 Molecular Medicine
Q2 Organic Chemistry
Q2 Pharmaceutical Science
2019
Kun, S.,
Kánya, N.,
Galó, N.,
Páhi, A.,
Mándi, A.,
Kurtán, T.,
Makleit, P.,
Veres, S.,
Sipos, Á.,
Docsa, T.,
Somsák, L.:
Glucopyranosylidene-spiro-benzo[b][1,4]oxazinones and -benzo[b][1,4]thiazinones: Synthesis and Investigation of Their Effects on Glycogen Phosphorylase and Plant Growth Inhibition.
J. Agric. Food Chem. 67 (24), 6884-6891, 2019.
Journal metrics:
Q1 Agricultural and Biological Sciences (miscellaneous)
Q1 Chemistry (miscellaneous)
Barr, D.,
Szennyes, E.,
Bokor, É.,
Al-Oanzi, Z.,
Moffatt, C.,
Kun, S.,
Docsa, T.,
Sipos, Á.,
Davies, M.,
Mathomes, R.,
Snape, T.,
Agius, L.,
Somsák, L.,
Hayes, J.:
Identification of C-[béta]-d-Glucopyranosyl Azole-Type Inhibitors of Glycogen Phosphorylase That Reduce Glycogenolysis in Hepatocytes: in Silico Design, Synthesis, in Vitro Kinetics, and ex Vivo Studies.
ACS Chem. Biol. 14 (7), 1460-1470, 2019.
Journal metrics:
Q1 Biochemistry
D1 Medicine (miscellaneous)
Q1 Molecular Medicine
Somsák, L.,
Bokor, É.,
Juhász, L.,
Kun, S.,
Lázár, L.,
Juhász-Tóth, É.,
Tóth, M.:
New syntheses towards C-glycosyl type glycomimetics.
Pure Appl. Chem. 91 (7), 1159-1175, 2019.
Journal metrics:
Q2 Chemical Engineering (miscellaneous)
Q2 Chemistry (miscellaneous)
Körhegyi, Z.,
Rózsa, D.,
Hajdu, I.,
Bodnár, M.,
Kertész, I.,
Kerekes, K.,
Kun, S.,
Kollár, J.,
Varga, J.,
Garai, I.,
Trencsényi, G.,
Borbély, J.:
Synthesis of 68Ga-Labeled Biopolymer-based Nanoparticle Imaging Agents for Positron-emission Tomography.
Anticancer Res. 39 (5), 2415-2427, 2019.
Journal metrics:
Q3 Cancer Research
Q2 Medicine (miscellaneous)
Q3 Oncology
2018
Kun, S.,
Begum, J.,
Kyriakis, E.,
Stamati, E.,
Barkas, T.,
Szennyes, E.,
Bokor, É.,
Szabó, E.,
Stravodimos, G.,
Sipos, Á.,
Docsa, T.,
Gergely, P.,
Moffatt, C.,
Patraskaki, M.,
Kokolaki, M.,
Gkerdi, A.,
Skamnaki, V.,
Leonidas, D.,
Somsák, L.,
Hayes, J.:
A multidisciplinary study of 3-(β-D-glucopyranosyl)-5-substituted-1,2,4-triazole derivatives as glycogen phosphorylase inhibitors: computation, synthesis, crystallography and kinetics reveal new potent inhibitors.
Eur. J. Med. Chem. 147 266-278, 2018.
Journal metrics:
Q1 Drug Discovery
Q1 Medicine (miscellaneous)
Q1 Organic Chemistry
Q1 Pharmacology
Nagy, L.,
Márton, J.,
Vida, A.,
Kis, G.,
Bokor, É.,
Kun, S.,
Gönczi, M.,
Docsa, T.,
Tóth, A.,
Antal, M.,
Gergely, P.,
Csóka, B.,
Pacher, P.,
Somsák, L.,
Bai, P.:
Glycogen phosphorylase inhibition improves beta cell function.
Br. J. Pharmacol. 175 (2), 301-319, 2018.
Kyriakis, E.,
Solovou, T.,
Kun, S.,
Czifrák, K.,
Szőcs, B.,
Juhász, L.,
Bokor, É.,
Stravodimos, G.,
Kantsadi, A.,
Chatzileontiadou, D.,
Skamnaki, V.,
Somsák, L.,
Leonidas, D.:
Probing the [beta]-pocket of the active site of human liver glycogen phosphorylase with 3-(C-[beta]-D-glucopyranosyl)-5-(4-substituted-phenyl)-1, 2, 4-triazole inhibitors.
Bioorganic Chem. 77 485-493, 2018.
Journal metrics:
Q3 Biochemistry
Q2 Drug Discovery
Q3 Molecular Biology
Q2 Organic Chemistry
Kun, S.,
Bokor, É.,
Sipos, Á.,
Docsa, T.,
Somsák, L.:
Synthesis of New C- and N-beta-D-Glucopyranosyl Derivatives of Imidazole, 1,2,3-Triazole and Tetrazole, and Their Evaluation as Inhibitors of Glycogen Phosphorylase.
Molecules. 23 (3), 1-17, 2018.
Journal metrics:
Q2 Analytical Chemistry
Q1 Chemistry (miscellaneous)
Q2 Drug Discovery
Q2 Medicine (miscellaneous)
Q3 Molecular Medicine
Q2 Organic Chemistry
Q1 Pharmaceutical Science
Q2 Physical and Theoretical Chemistry
2017
Bokor, É.,
Kun, S.,
Goyard, D.,
Tóth, M.,
Praly, J.,
Vidal, S.,
Somsák, L.:
C-Glycopyranosyl Arenes and Hetarenes: Synthetic Methods and Bioactivity Focused on Antidiabetic Potential.
Chem. Rev. 117 (3), 1687-1764, 2017.
Journal metrics:
D1 Chemistry (miscellaneous)
Szabó, E.,
Kun, S.,
Mándi, A.,
Kurtán, T.,
Somsák, L.:
Glucopyranosylidene-Spiro-Thiazolinones: Synthetic Studies and Determination of Absolute Configuration by TDDFT-ECD Calculations.
Molecules. 22 (10), 1760-1774, 2017.
Journal metrics:
Q1 Analytical Chemistry
Q1 Chemistry (miscellaneous)
Q2 Drug Discovery
Q2 Medicine (miscellaneous)
Q3 Molecular Medicine
Q2 Organic Chemistry
Q1 Pharmaceutical Science
Q2 Physical and Theoretical Chemistry
Kantsadi, A.,
Stravodimos, G.,
Kyriakis, E.,
Chatzileontiadou, D.,
Solovou, T.,
Kun, S.,
Bokor, É.,
Somsák, L.:
van der Waals interactions govern C-[beta]-D-glucopyranosyl triazoles' nM inhibitory potency in human liver glycogen phosphorylase.
J. Struct. Biol. 199 (1), 57-67, 2017.
2016
Kantsadi, A.,
Bokor, É.,
Kun, S.,
Stravodimos, G.,
Chatzileontiadou, D.,
Leonidas, D.,
Juhász-Tóth, É.,
Szakács, A.,
Batta, G.,
Docsa, T.,
Gergely, P.,
Somsák, L.:
Synthetic, enzyme kinetic, and protein crystallographic studies of C-[béta]-D-glucopyranosyl pyrroles and imidazoles reveal and explain low nanomolar inhibition of human liver glycogen phosphorylase.
Eur. J. Med. Chem. 123 737-745, 2016.
Journal metrics:
Q1 Drug Discovery
Q1 Medicine (miscellaneous)
Q1 Organic Chemistry
Q1 Pharmacology
2015
Bokor, É.,
Kun, S.,
Docsa, T.,
Gergely, P.,
Somsák, L.:
4(5)-Aryl-2-C-glucopyranosyl-imidazoles as New Nanomolar Glucose Analogue Inhibitors of Glycogen Phosphorylase.
ACS Med. Chem. Lett. 6 1215-1219, 2015.
Journal metrics:
Q2 Biochemistry
Q1 Drug Discovery
Q1 Organic Chemistry
Misra, A.,
Bokor, É.,
Kun, S.,
Bolyog-Nagy, E.,
Kathó, Á.,
Joó, F.,
Somsák, L.:
Chemoselective hydration of glycosyl cyanides to C-glycosyl formamides using ruthenium complexes in aqueous media.
Tetrahedron Lett. 56 (44), 5995-5998, 2015.
Journal metrics:
Q3 Biochemistry
Q2 Drug Discovery
Q2 Organic Chemistry
2014
Kun, S.,
Bokor, É.,
Varga, G.,
Szőcs, B.,
Páhi, A.,
Czifrák, K.,
Tóth, M.,
Juhász, L.,
Docsa, T.,
Gergely, P.,
Somsák, L.:
New synthesis of 3-(β-D-glucopyranosyl)-5-substituted-1,2,4- triazoles, nanomolar inhibitors of glycogen phosphorylase.
Eur. J. Med. Chem. 76 567-579, 2014.
Journal metrics:
Q1 Drug Discovery
Q1 Medicine (miscellaneous)
Q1 Organic Chemistry
Q1 Pharmacology
Somsák, L.,
Bokor, É.,
Czibere, B.,
Czifrák, K.,
Koppány, C.,
Kulcsár, L.,
Kun, S.,
Szilágyi, E.,
Tóth, M.,
Docsa, T.,
Gergely, P.:
Synthesis of C-xylopyranosyl- and xylopyranosylidene-spiro-heterocycles as potential inhibitors of glycogen phosphorylase.
Carbohydr. Res. 399 38-48, 2014.
Journal metrics:
Q2 Analytical Chemistry
Q3 Biochemistry
Q2 Medicine (miscellaneous)
Q2 Organic Chemistry
2023
Kun, S.,
Mathomes, R.,
Docsa, T.,
Somsák, L.,
Hayes, J.:
Design and Synthesis of 3-(β-D-Glucopyranosyl)-4-amino/4-guanidino Pyrazole Derivatives and Analysis of Their Glycogen Phosphorylase Inhibitory Potential.
Molecules. 28 (7), 1-19, 2023.
Journal metrics:
Q1 Analytical Chemistry
Q1 Chemistry (miscellaneous)
Q2 Drug Discovery
Q2 Medicine (miscellaneous)
Q3 Molecular Medicine
Q2 Organic Chemistry
Q1 Pharmaceutical Science
Q2 Physical and Theoretical Chemistry
2022
2021
Sipos, Á.,
Szennyes, E.,
Hajnal, É.,
Kun, S.,
Szabó, E.,
Uray, K.,
Somsák, L.,
Docsa, T.,
Bokor, É.:
Dual-Target Compounds against Type 2 Diabetes Mellitus: proof of Concept for Sodium Dependent Glucose Transporter (SGLT) and Glycogen Phosphorylase (GP) Inhibitors.
Pharmaceuticals. 14 (4), 1-27, 2021.
Journal metrics:
Q1 Drug Discovery
Q2 Molecular Medicine
Q1 Pharmaceutical Science
Tsagkarakou, A.,
Chasapi, S.,
Koulas, S.,
Tsialtas, I.,
Kyriakis, E.,
Drakou, C.,
Kun, S.,
Somsák, L.,
Spyroulias, G.,
Psarra, A.,
Leonidas, D.:
Structure activity relationship of the binding of p-coumaroyl glucose to glycogen phosphorylase and its effect on hepatic cell metabolic pathways.
European Journal of Medicinal Chemistry Reports. 3 1-11, 2021.
2020
Gorliczay, E.,
Tamás, J.,
Kun, S.,
Huzsvai, L.,
Bárány, L.:
Examination and statistical evaluation of physico-chemical parameters of windrow composting.
Agrártud. Közl. 1 33-38, 2020.
Kiss, N.,
Nagy, P.,
Tóth, F.,
Gorliczay, E.,
Madar, L.,
Kun, S.,
Tamás, J.:
Improving the water management properties of different soil type.
In: A klímaváltozás kihívásai a következő évtizedekben : előadások kivonatai, Szent István Egyetem, Keszthely, 54, 2020.
Kyriakis, E.,
Karra, A.,
Papaioannou, O.,
Solovou, T.,
Skamnaki, V.,
Liggri, P.,
Zographos, S.,
Szennyes, E.,
Bokor, É.,
Kun, S.,
Psarra, A.,
Somsák, L.,
Leonidas, D.:
The architecture of hydrogen and sulfur α-hole interactions explain differences in the inhibitory potency of C-β-d-glucopyranosyl thiazoles, imidazoles and an N-β-d glucopyranosyl tetrazole for human liver glycogen phosphorylase and offer new insights to structure-based design.
Bioorg. Med. Chem. 28 (1), 1-10, 2020.
Journal metrics:
Q3 Biochemistry
Q2 Clinical Biochemistry
Q2 Drug Discovery
Q3 Molecular Biology
Q3 Molecular Medicine
Q2 Organic Chemistry
Q2 Pharmaceutical Science
2019
Kun, S.,
Kánya, N.,
Galó, N.,
Páhi, A.,
Mándi, A.,
Kurtán, T.,
Makleit, P.,
Veres, S.,
Sipos, Á.,
Docsa, T.,
Somsák, L.:
Glucopyranosylidene-spiro-benzo[b][1,4]oxazinones and -benzo[b][1,4]thiazinones: Synthesis and Investigation of Their Effects on Glycogen Phosphorylase and Plant Growth Inhibition.
J. Agric. Food Chem. 67 (24), 6884-6891, 2019.
Journal metrics:
Q1 Agricultural and Biological Sciences (miscellaneous)
Q1 Chemistry (miscellaneous)
Barr, D.,
Szennyes, E.,
Bokor, É.,
Al-Oanzi, Z.,
Moffatt, C.,
Kun, S.,
Docsa, T.,
Sipos, Á.,
Davies, M.,
Mathomes, R.,
Snape, T.,
Agius, L.,
Somsák, L.,
Hayes, J.:
Identification of C-[béta]-d-Glucopyranosyl Azole-Type Inhibitors of Glycogen Phosphorylase That Reduce Glycogenolysis in Hepatocytes: in Silico Design, Synthesis, in Vitro Kinetics, and ex Vivo Studies.
ACS Chem. Biol. 14 (7), 1460-1470, 2019.
Journal metrics:
Q1 Biochemistry
D1 Medicine (miscellaneous)
Q1 Molecular Medicine
Somsák, L.,
Bokor, É.,
Juhász, L.,
Kun, S.,
Lázár, L.,
Juhász-Tóth, É.,
Tóth, M.:
New syntheses towards C-glycosyl type glycomimetics.
Pure Appl. Chem. 91 (7), 1159-1175, 2019.
Journal metrics:
Q2 Chemical Engineering (miscellaneous)
Q2 Chemistry (miscellaneous)
Körhegyi, Z.,
Rózsa, D.,
Hajdu, I.,
Bodnár, M.,
Kertész, I.,
Kerekes, K.,
Kun, S.,
Kollár, J.,
Varga, J.,
Garai, I.,
Trencsényi, G.,
Borbély, J.:
Synthesis of 68Ga-Labeled Biopolymer-based Nanoparticle Imaging Agents for Positron-emission Tomography.
Anticancer Res. 39 (5), 2415-2427, 2019.
Journal metrics:
Q3 Cancer Research
Q2 Medicine (miscellaneous)
Q3 Oncology
2018
Kun, S.,
Begum, J.,
Kyriakis, E.,
Stamati, E.,
Barkas, T.,
Szennyes, E.,
Bokor, É.,
Szabó, E.,
Stravodimos, G.,
Sipos, Á.,
Docsa, T.,
Gergely, P.,
Moffatt, C.,
Patraskaki, M.,
Kokolaki, M.,
Gkerdi, A.,
Skamnaki, V.,
Leonidas, D.,
Somsák, L.,
Hayes, J.:
A multidisciplinary study of 3-(β-D-glucopyranosyl)-5-substituted-1,2,4-triazole derivatives as glycogen phosphorylase inhibitors: computation, synthesis, crystallography and kinetics reveal new potent inhibitors.
Eur. J. Med. Chem. 147 266-278, 2018.
Journal metrics:
Q1 Drug Discovery
Q1 Medicine (miscellaneous)
Q1 Organic Chemistry
Q1 Pharmacology
Nagy, L.,
Márton, J.,
Vida, A.,
Kis, G.,
Bokor, É.,
Kun, S.,
Gönczi, M.,
Docsa, T.,
Tóth, A.,
Antal, M.,
Gergely, P.,
Csóka, B.,
Pacher, P.,
Somsák, L.,
Bai, P.:
Glycogen phosphorylase inhibition improves beta cell function.
Br. J. Pharmacol. 175 (2), 301-319, 2018.
Kyriakis, E.,
Solovou, T.,
Kun, S.,
Czifrák, K.,
Szőcs, B.,
Juhász, L.,
Bokor, É.,
Stravodimos, G.,
Kantsadi, A.,
Chatzileontiadou, D.,
Skamnaki, V.,
Somsák, L.,
Leonidas, D.:
Probing the [beta]-pocket of the active site of human liver glycogen phosphorylase with 3-(C-[beta]-D-glucopyranosyl)-5-(4-substituted-phenyl)-1, 2, 4-triazole inhibitors.
Bioorganic Chem. 77 485-493, 2018.
Journal metrics:
Q3 Biochemistry
Q2 Drug Discovery
Q3 Molecular Biology
Q2 Organic Chemistry
Kun, S.,
Bokor, É.,
Sipos, Á.,
Docsa, T.,
Somsák, L.:
Synthesis of New C- and N-beta-D-Glucopyranosyl Derivatives of Imidazole, 1,2,3-Triazole and Tetrazole, and Their Evaluation as Inhibitors of Glycogen Phosphorylase.
Molecules. 23 (3), 1-17, 2018.
Journal metrics:
Q2 Analytical Chemistry
Q1 Chemistry (miscellaneous)
Q2 Drug Discovery
Q2 Medicine (miscellaneous)
Q3 Molecular Medicine
Q2 Organic Chemistry
Q1 Pharmaceutical Science
Q2 Physical and Theoretical Chemistry
2017
Bokor, É.,
Kun, S.,
Goyard, D.,
Tóth, M.,
Praly, J.,
Vidal, S.,
Somsák, L.:
C-Glycopyranosyl Arenes and Hetarenes: Synthetic Methods and Bioactivity Focused on Antidiabetic Potential.
Chem. Rev. 117 (3), 1687-1764, 2017.
Journal metrics:
D1 Chemistry (miscellaneous)
Szabó, E.,
Kun, S.,
Mándi, A.,
Kurtán, T.,
Somsák, L.:
Glucopyranosylidene-Spiro-Thiazolinones: Synthetic Studies and Determination of Absolute Configuration by TDDFT-ECD Calculations.
Molecules. 22 (10), 1760-1774, 2017.
Journal metrics:
Q1 Analytical Chemistry
Q1 Chemistry (miscellaneous)
Q2 Drug Discovery
Q2 Medicine (miscellaneous)
Q3 Molecular Medicine
Q2 Organic Chemistry
Q1 Pharmaceutical Science
Q2 Physical and Theoretical Chemistry
Kantsadi, A.,
Stravodimos, G.,
Kyriakis, E.,
Chatzileontiadou, D.,
Solovou, T.,
Kun, S.,
Bokor, É.,
Somsák, L.:
van der Waals interactions govern C-[beta]-D-glucopyranosyl triazoles' nM inhibitory potency in human liver glycogen phosphorylase.
J. Struct. Biol. 199 (1), 57-67, 2017.
2016
Kantsadi, A.,
Bokor, É.,
Kun, S.,
Stravodimos, G.,
Chatzileontiadou, D.,
Leonidas, D.,
Juhász-Tóth, É.,
Szakács, A.,
Batta, G.,
Docsa, T.,
Gergely, P.,
Somsák, L.:
Synthetic, enzyme kinetic, and protein crystallographic studies of C-[béta]-D-glucopyranosyl pyrroles and imidazoles reveal and explain low nanomolar inhibition of human liver glycogen phosphorylase.
Eur. J. Med. Chem. 123 737-745, 2016.
Journal metrics:
Q1 Drug Discovery
Q1 Medicine (miscellaneous)
Q1 Organic Chemistry
Q1 Pharmacology
2015
Bokor, É.,
Kun, S.,
Docsa, T.,
Gergely, P.,
Somsák, L.:
4(5)-Aryl-2-C-glucopyranosyl-imidazoles as New Nanomolar Glucose Analogue Inhibitors of Glycogen Phosphorylase.
ACS Med. Chem. Lett. 6 1215-1219, 2015.
Journal metrics:
Q2 Biochemistry
Q1 Drug Discovery
Q1 Organic Chemistry
Misra, A.,
Bokor, É.,
Kun, S.,
Bolyog-Nagy, E.,
Kathó, Á.,
Joó, F.,
Somsák, L.:
Chemoselective hydration of glycosyl cyanides to C-glycosyl formamides using ruthenium complexes in aqueous media.
Tetrahedron Lett. 56 (44), 5995-5998, 2015.
Journal metrics:
Q3 Biochemistry
Q2 Drug Discovery
Q2 Organic Chemistry
2014
Kun, S.,
Bokor, É.,
Varga, G.,
Szőcs, B.,
Páhi, A.,
Czifrák, K.,
Tóth, M.,
Juhász, L.,
Docsa, T.,
Gergely, P.,
Somsák, L.:
New synthesis of 3-(β-D-glucopyranosyl)-5-substituted-1,2,4- triazoles, nanomolar inhibitors of glycogen phosphorylase.
Eur. J. Med. Chem. 76 567-579, 2014.
Journal metrics:
Q1 Drug Discovery
Q1 Medicine (miscellaneous)
Q1 Organic Chemistry
Q1 Pharmacology
Somsák, L.,
Bokor, É.,
Czibere, B.,
Czifrák, K.,
Koppány, C.,
Kulcsár, L.,
Kun, S.,
Szilágyi, E.,
Tóth, M.,
Docsa, T.,
Gergely, P.:
Synthesis of C-xylopyranosyl- and xylopyranosylidene-spiro-heterocycles as potential inhibitors of glycogen phosphorylase.
Carbohydr. Res. 399 38-48, 2014.
Journal metrics:
Q2 Analytical Chemistry
Q3 Biochemistry
Q2 Medicine (miscellaneous)
Q2 Organic Chemistry
2012
Tóth, M.,
Kun, S.,
Somsák, L.,
Goyard, D.:
Preparation of exo-Glycals from 2,6-Anhydro-aldose-tosylhydrazones.
In: Carbohydrate Chemistry : Proven Synthetic Methods Vol. 1.. Ed.: Pavol Kováč, CRC Press, Boca Raton, 367-375, 2012. ISBN: 9781439866894
2011
Kun, S.,
Nagy, G.,
Tóth, M.,
Czecze, L.,
Van Nhien, A.,
Docsa, T.,
Gergely, P.,
Charavgi, M.,
Skourti, P.,
Chrysina, E.,
Patonay, T.,
Somsák, L.:
Synthesis of variously coupled conjugates of d-glucose, 1,3,4-oxadiazole, and 1,2,3-triazole for inhibition of glycogen phosphorylase.
Carbohydr. Res. 346 (12), 1427-1438, 2011.
Journal metrics:
Q2 Analytical Chemistry
Q3 Biochemistry
Q2 Medicine (miscellaneous)
Q2 Organic Chemistry
2010
Somsák, L.,
Bokor, É.,
Czifrák, K.,
Kónya, B.,
Kun, S.,
Tóth, M.:
A glikogén foszforiláz glükózanalóg gátlószerei, mint potenciális antidiabetikumok.
Magy. Kém. F. 116 (1), 19-30, 2010.
2009
Tóth, M.,
Kun, S.,
Bokor, É.,
Benltifa, M.,
Tallec, G.,
Vidal, S.,
Docsa, T.,
Gergely, P.,
Somsák, L.,
Praly, J.:
Synthesis and structure-activity relationships of C-glycosylated oxadiazoles as inhibitors of glycogen phosphorylase.
Bioorg. Med. Chem. 17 (13), 4773-4785, 2009.
Journal metrics:
Q2 Biochemistry
Q1 Clinical Biochemistry
Q1 Drug Discovery
Q3 Molecular Biology
Q2 Molecular Medicine
Q1 Organic Chemistry
Q1 Pharmaceutical Science
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updated: 2024-12-19, 02:04