Összes letöltés a DEA-ból: 5469
country | downloads |
---|---|
United States (US) | 2984 |
China (CN) | 437 |
Hong Kong S.A.R., China (HK) | 394 |
Germany (DE) | 216 |
France (FR) | 137 |
United Kingdom (GB) | 131 |
Hungary (HU) | 112 |
Russia (RU) | 101 |
Sweden (SE) | 94 |
Netherlands (NL) | 73 |
India (IN) | 71 |
Ireland (IE) | 56 |
Indonesia (ID) | 41 |
Singapore (SG) | 41 |
Japan (JP) | 25 |
Canada (CA) | 24 |
Czech Republic (CZ) | 23 |
Turkey (TR) | 22 |
Finland (FI) | 21 |
Australia (AU) | 17 |
South Africa (ZA) | 17 |
Pakistan (PK) | 16 |
Philippines (PH) | 15 |
Vietnam (VN) | 14 |
Lithuania (LT) | 13 |
Brazil (BR) | 11 |
Ukraine (UA) | 11 |
Poland (PL) | 10 |
Morocco (MA) | 9 |
Romania (RO) | 9 |
Chile (CL) | 8 |
Greece (GR) | 8 |
Macao S.A.R., China (MO) | 8 |
Spain (ES) | 7 |
Egypt (EG) | 6 |
Iraq (IQ) | 5 |
Italy (IT) | 4 |
Thailand (TH) | 4 |
United Arab Emirates (AE) | 3 |
Austria (AT) | 3 |
Mexico (MX) | 3 |
Norway (NO) | 3 |
Saudi Arabia (SA) | 3 |
Belgium (BE) | 2 |
Bulgaria (BG) | 2 |
Belarus (BY) | 2 |
Switzerland (CH) | 2 |
Luxembourg (LU) | 2 |
Malaysia (MY) | 2 |
Nigeria (NG) | 2 |
Slovakia (SK) | 2 |
Tunisia (TN) | 2 |
Benin (BJ) | 1 |
Denmark (DK) | 1 |
Algeria (DZ) | 1 |
Estonia (EE) | 1 |
Ghana (GH) | 1 |
Croatia (HR) | 1 |
Martinique (MQ) | 1 |
Mauritius (MU) | 1 |
Puerto Rico (PR) | 1 |
Portugal (PT) | 1 |
Syria (SY) | 1 |
n.a. | 230 |
Megjelenés | Publication | Fájlletöltések |
---|---|---|
2024 | Homolya, L., Mathomes, R., Varga, L., Docsa, T., Juhász, L., Hayes, J., Somsák, L.: Synthesis, in silico and kinetics evaluation of N-(beta-D-glucopyranosyl)-2-arylimidazole-4(5)-carboxamides and N-(beta-D-glucopyranosyl)-4(5)-arylimidazole-2-carboxamides as glycogen phosphorylase inhibitors. Int. J. Mol. Sci. 25 (9), 1-21, 2024. Teljes szöveg: https://hdl.handle.net/2437/369417 Folyóirat-mutatók:
Q2 Catalysis (2023) Q1 Computer Science Applications (2023) D1 Inorganic Chemistry (2023) Q1 Medicine (miscellaneous) (2023) Q2 Molecular Biology (2023) D1 Organic Chemistry (2023) Q1 Physical and Theoretical Chemistry (2023) D1 Spectroscopy (2023) | Kiadói változat: 17 |
2023 | Kun, S., Mathomes, R., Docsa, T., Somsák, L., Hayes, J.: Design and Synthesis of 3-(β-D-Glucopyranosyl)-4-amino/4-guanidino Pyrazole Derivatives and Analysis of Their Glycogen Phosphorylase Inhibitory Potential. Molecules. 28 (7), 1-19, 2023. Teljes szöveg: https://hdl.handle.net/2437/348528 Folyóirat-mutatók:
Q1 Analytical Chemistry Q1 Chemistry (miscellaneous) Q2 Drug Discovery Q2 Medicine (miscellaneous) Q3 Molecular Medicine Q2 Organic Chemistry Q1 Pharmaceutical Science Q2 Physical and Theoretical Chemistry | kiadói változat: 9 |
2023 | Kola, J., Docsa, T., Uray, K.: Mechanosensing in the Physiology and Pathology of the Gastrointestinal Tract. Int. J. Mol. Sci. 24 (1), 1-12, 2023. Teljes szöveg: https://hdl.handle.net/2437/355721 Folyóirat-mutatók:
Q2 Catalysis Q1 Computer Science Applications D1 Inorganic Chemistry Q1 Medicine (miscellaneous) Q2 Molecular Biology D1 Organic Chemistry Q1 Physical and Theoretical Chemistry D1 Spectroscopy | kiadói változat: 6 |
2023 | Kola, J., Turarova, B., Csige, D., Sipos, Á., Varga, L., Gergely, B., Refai, F., Uray, I., Docsa, T., Uray, K.: Stretch-Induced Down-Regulation of HCN2 Suppresses Contractile Activity. Molecules. 28 (11), 1-14, 2023. Teljes szöveg: https://hdl.handle.net/2437/354369 Folyóirat-mutatók:
Q1 Analytical Chemistry Q1 Chemistry (miscellaneous) Q2 Drug Discovery Q2 Medicine (miscellaneous) Q3 Molecular Medicine Q2 Organic Chemistry Q1 Pharmaceutical Science Q2 Physical and Theoretical Chemistry | kiadói változat: 19 |
2022 | Docsa, T., Sipos, Á., Cox, C., Uray, K.: The Role of Inflammatory Mediators in the Development of Gastrointestinal Motility Disorders. Int. J. Mol. Sci. 23 (13), 1-22, 2022. Teljes szöveg: https://hdl.handle.net/2437/335880 Folyóirat-mutatók:
Q2 Catalysis Q1 Computer Science Applications D1 Inorganic Chemistry Q1 Medicine (miscellaneous) Q2 Molecular Biology Q1 Organic Chemistry Q1 Physical and Theoretical Chemistry D1 Spectroscopy | kiadói változat: 26 |
2021 | Sipos, Á., Szennyes, E., Hajnal, É., Kun, S., Szabó, E., Uray, K., Somsák, L., Docsa, T., Bokor, É.: Dual-Target Compounds against Type 2 Diabetes Mellitus: proof of Concept for Sodium Dependent Glucose Transporter (SGLT) and Glycogen Phosphorylase (GP) Inhibitors. Pharmaceuticals. 14 (4), 1-27, 2021. Teljes szöveg: https://hdl.handle.net/2437/305911 Folyóirat-mutatók:
Q1 Drug Discovery Q2 Molecular Medicine Q1 Pharmaceutical Science | kiadói változat: 28 |
2020 | Docsa, T., Bhattarai, D., Sipos, Á., Wade, C., Cox, C., Uray, K.: CXCL1 is upregulated during the development of ileus resulting in decreased intestinal contractile activity. Neurogastroenterol. Motil. 32 (3), 1-12, 2020. Teljes szöveg: https://hdl.handle.net/2437/281431 Folyóirat-mutatók:
Q2 Endocrine and Autonomic Systems Q1 Gastroenterology Q1 Physiology | kiadói változat: 72 |
2020 | Nagy, L., Béke, F., Juhász, L., Kovács, T., Juhász-Tóth, É., Docsa, T., Tóth, A., Gergely, P., Somsák, L., Bai, P.: Glycogen phosphorylase inhibitor, 2,3-bis[(2E)-3-(4-hydroxyphenyl)prop-2-enamido] butanedioic acid (BF142), improves baseline insulin secretion of MIN6 insulinoma cells. PLoS One. 15 (9), 1-15, 2020. Teljes szöveg: https://hdl.handle.net/2437/291701 Folyóirat-mutatók:
D1 Multidisciplinary | post-print: 37 kiadói változat: 21 |
2018 | Nagy, L., Márton, J., Vida, A., Kis, G., Bokor, É., Kun, S., Gönczi, M., Docsa, T., Tóth, A., Antal, M., Gergely, P., Csóka, B., Pacher, P., Somsák, L., Bai, P.: Glycogen phosphorylase inhibition improves beta cell function. Br. J. Pharmacol. 175 (2), 301-319, 2018. Teljes szöveg: https://hdl.handle.net/2437/236466 Folyóirat-mutatók:
D1 Pharmacology | pre-print: 101 |
2016 | Bokor, É., Széles, Z., Docsa, T., Gergely, P., Somsák, L.: C-Glucopyranosyl-1,2,4-triazol-5-ones: synthesis and inhibition of glycogen phosphorylase. Carbohydr. Res. 429 128-134, 2016. Teljes szöveg: https://hdl.handle.net/2437/228291 Folyóirat-mutatók:
Q2 Analytical Chemistry Q3 Biochemistry Q2 Medicine (miscellaneous) Q2 Organic Chemistry | post-print: 162 |
2016 | Goyard, D., Kónya, B., Chajistamatiou, A., Chrysina, E., Leroy, J., Balzarin, S., Tournier, M., Tousch, D., Petit, P., Duret, C., Maurel, P., Somsák, L., Docsa, T., Gergely, P., Praly, J., Azay-Milhau, J., Vidal, S.: Glucose-derived spiro-isoxazolines are anti-hyperglycemic agents against type 2 diabetes through glycogen phosphorylase inhibition. Eur. J. Med. Chem. 108 444-454, 2016. Teljes szöveg: https://hdl.handle.net/2437/221468 Folyóirat-mutatók:
Q1 Drug Discovery Q1 Medicine (miscellaneous) Q1 Organic Chemistry Q1 Pharmacology | post-print: 672 |
2016 | Szennyes, E., Bokor, É., Batta, G., Docsa, T., Gergely, P., Somsák, L.: Improved preparation of 4(5)-aryl-2-(β-D-glucopyranosyl)-imidazoles, the most efficient glucose analogue inhibitors of glycogen phosphorylase. RSC Adv. 6 (97), 94787-94794, 2016. Teljes szöveg: https://hdl.handle.net/2437/230831 Folyóirat-mutatók:
Q1 Chemical Engineering (miscellaneous) Q1 Chemistry (miscellaneous) | Kiadói változat: 153 |
2016 | Petrušová, M., Smrtičová, H., Pribulová, B., Vlčková, S., Uhliariková, I., Docsa, T., Somsák, L., Petruš, L.: One pot InCl3-catalyzed synthesis of 1-glycosylmethyl-1H-imidazoles. Tetrahedron. 72 (17), 2116-2121, 2016. Teljes szöveg: https://hdl.handle.net/2437/225481 Folyóirat-mutatók:
Q2 Biochemistry Q2 Drug Discovery Q2 Organic Chemistry | post-print: 103 |
2016 | Kantsadi, A., Bokor, É., Kun, S., Stravodimos, G., Chatzileontiadou, D., Leonidas, D., Juhász-Tóth, É., Szakács, A., Batta, G., Docsa, T., Gergely, P., Somsák, L.: Synthetic, enzyme kinetic, and protein crystallographic studies of C-[béta]-D-glucopyranosyl pyrroles and imidazoles reveal and explain low nanomolar inhibition of human liver glycogen phosphorylase. Eur. J. Med. Chem. 123 737-745, 2016. Teljes szöveg: https://hdl.handle.net/2437/229840 Folyóirat-mutatók:
Q1 Drug Discovery Q1 Medicine (miscellaneous) Q1 Organic Chemistry Q1 Pharmacology | pre-print: 194 |
2015 | Donnier-Maréchal, M., Goyard, D., Folliard, V., Docsa, T., Gergely, P., Praly, J., Vidal, S.: 3-Glucosylated 5-amino-1,2,4-oxadiazoles: synthesis and evaluation as glycogen phosphorylase inhibitors. Beilstein J. Org. Chem. 11 499-503, 2015. Teljes szöveg: https://hdl.handle.net/2437/209870 Folyóirat-mutatók:
Q1 Organic Chemistry | kiadói változat: 59 |
2015 | Bokor, É., Szennyes, E., Csupász, T., Tóth, N., Docsa, T., Gergely, P., Somsák, L.: C-(2-Deoxy-D-arabino-hex-1-enopyranosyl)-oxadiazoles: synthesis of possible isomers and their evaluation as glycogen phosphorylase inhibitors. Carbohydr. Res. 412 71-79, 2015. Teljes szöveg: https://hdl.handle.net/2437/214559 Folyóirat-mutatók:
Q2 Analytical Chemistry Q3 Biochemistry Q2 Medicine (miscellaneous) Q2 Organic Chemistry | post-print: 174 |
2015 | Begum, J., Varga, G., Docsa, T., Gergely, P., Hayes, J., Juhász, L., Somsák, L.: Computationally motivated synthesis and enzyme kinetic evaluation of N-([beta]-D-glucopyranosyl)-1,2,4-triazolecarboxamides as glycogen phosphorylase inhibitors. Med. Chem. Commun. 6 (1), 80-89, 2015. Teljes szöveg: https://hdl.handle.net/2437/203139 Folyóirat-mutatók:
Q2 Biochemistry Q1 Pharmaceutical Science | post-print: 124 |
2015 | Goyard, D., Docsa, T., Gergely, P., Praly, J., Vidal, S.: Synthesis of 4-amidomethyl-1-glucosyl-1,2,3-triazoles and evaluation as glycogen phosphorylase inhibitors. Carbohydr. Res. 402 245-251, 2015. Teljes szöveg: https://hdl.handle.net/2437/203107 Folyóirat-mutatók:
Q2 Analytical Chemistry Q3 Biochemistry Q2 Medicine (miscellaneous) Q2 Organic Chemistry | pre-print: 146 |
2014 | Czifrák, K., Páhi, A., Deák, S., Kiss-Szikszai, A., Kövér, K., Docsa, T., Gergely, P., Alexacou, K., Papakonstantinou, M., Leonidas, D., Zographos, S., Chrysina, E., Somsák, L.: Glucopyranosylidene-spiro-iminothiazolidinone, a New Bicyclic Ring System: Synthesis, Derivatization, and Evaluation for Inhibition of Glycogen Phosphorylase by Enzyme Kinetic and Crystallographic Methods. Bioorg. Med. Chem. 22 (15), 4028-4041, 2014. Teljes szöveg: https://hdl.handle.net/2437/194534 Folyóirat-mutatók:
Q2 Biochemistry Q2 Clinical Biochemistry Q1 Drug Discovery Q3 Molecular Biology Q2 Molecular Medicine Q1 Organic Chemistry Q1 Pharmaceutical Science | post-print: 267 |
2014 | Kun, S., Bokor, É., Varga, G., Szőcs, B., Páhi, A., Czifrák, K., Tóth, M., Juhász, L., Docsa, T., Gergely, P., Somsák, L.: New synthesis of 3-(β-D-glucopyranosyl)-5-substituted-1,2,4- triazoles, nanomolar inhibitors of glycogen phosphorylase. Eur. J. Med. Chem. 76 567-579, 2014. Teljes szöveg: https://hdl.handle.net/2437/181459 Folyóirat-mutatók:
Q1 Drug Discovery Q1 Medicine (miscellaneous) Q1 Organic Chemistry Q1 Pharmacology | post-print: 203 |
2014 | Somsák, L., Bokor, É., Czibere, B., Czifrák, K., Koppány, C., Kulcsár, L., Kun, S., Szilágyi, E., Tóth, M., Docsa, T., Gergely, P.: Synthesis of C-xylopyranosyl- and xylopyranosylidene-spiro-heterocycles as potential inhibitors of glycogen phosphorylase. Carbohydr. Res. 399 38-48, 2014. Teljes szöveg: https://hdl.handle.net/2437/201184 Folyóirat-mutatók:
Q2 Analytical Chemistry Q3 Biochemistry Q2 Medicine (miscellaneous) Q2 Organic Chemistry | post-print: 249 |
2013 | Bokor, É., Docsa, T., Gergely, P., Somsák, L.: C-Glucopyranosyl-1,2,4-triazoles As New Potent Inhibitors of Glycogen Phosphorylase. ACS Med. Chem. Lett. 4 (7), 612-615, 2013. Teljes szöveg: https://hdl.handle.net/2437/172417 Folyóirat-mutatók:
Q1 Biochemistry Q1 Drug Discovery Q1 Organic Chemistry | post-print: 108 |
2013 | Nagy, L., Docsa, T., Szántó, M., Brunyánszki, A., Hegedűs, C., Márton, J., Kónya, B., Virág, L., Somsák, L., Gergely, P., Bai, P.: Glycogen Phosphorylase Inhibitor N-(3,5-Dimethyl-Benzoyl)-N'-(β-D-Glucopyranosyl)Urea Improves Glucose Tolerance under Normoglycemic and Diabetic Conditions and Rearranges Hepatic Metabolism. PLoS One. 8 (7), e69420-, 2013. Teljes szöveg: https://hdl.handle.net/2437/172283 Folyóirat-mutatók:
D1 Agricultural and Biological Sciences (miscellaneous) Q1 Biochemistry, Genetics and Molecular Biology (miscellaneous) D1 Medicine (miscellaneous) | kiadói változat: 105 |
2013 | Polyák, M., Varga, G., Szilágyi, B., Juhász, L., Docsa, T., Gergely, P., Begum, J., Hayes, J., Somsák, L.: Synthesis, enzyme kinetics and computational evaluation of N-(β-d-glucopyranosyl) oxadiazolecarboxamides as glycogen phosphorylase inhibitors. Bioorg. Med. Chem. 21 (18), 5738-5747, 2013. Teljes szöveg: https://hdl.handle.net/2437/172418 Folyóirat-mutatók:
Q2 Biochemistry Q2 Clinical Biochemistry Q1 Drug Discovery Q3 Molecular Biology Q2 Molecular Medicine Q1 Organic Chemistry Q1 Pharmaceutical Science | post-print: 247 |
2013 | Szőcs, B., Tóth, M., Docsa, T., Gergely, P., Somsák, L.: Synthesis of 2-(β-D-glucopyranosyl)-5-(substituted-amino)-1,3,4-oxa-and -thiadiazoles for the inhibition of glycogen phosphorylase. Carbohydr. Res. 381C 187-195, 2013. Teljes szöveg: https://hdl.handle.net/2437/174243 Folyóirat-mutatók:
Q2 Analytical Chemistry Q3 Biochemistry Q2 Medicine (miscellaneous) Q2 Organic Chemistry | post-print: 229 |
2013 | Tóth, M., Szőcs, B., Kaszás, T., Docsa, T., Gergely, P., Somsák, L.: Synthesis of 2-(β-D-glucopyranosylamino)-5-substituted-1,3,4-oxadiazoles for inhibition of glycogen phosphorylase. Carbohydr. Res. 381C 196-204, 2013. Teljes szöveg: https://hdl.handle.net/2437/174244 Folyóirat-mutatók:
Q2 Analytical Chemistry Q3 Biochemistry Q2 Medicine (miscellaneous) Q2 Organic Chemistry | post-print: 133 |
2013 | Bokor, É., Szilágyi, E., Docsa, T., Gergely, P., Somsák, L.: Synthesis of substituted 2-(β-d-glucopyranosyl)-benzimidazoles and their evaluation as inhibitors of glycogen phosphorylase. Carbohydr. Res. 381C 179-186, 2013. Teljes szöveg: https://hdl.handle.net/2437/174234 Folyóirat-mutatók:
Q2 Analytical Chemistry Q3 Biochemistry Q2 Medicine (miscellaneous) Q2 Organic Chemistry | post-print: 170 |
2013 | Varga, G., Docsa, T., Gergely, P., Juhász, L., Somsák, L.: Synthesis of tartaric acid analogues of FR258900 and their evaluation as glycogen phosphorylase inhibitors. Bioorg. Med. Chem. Lett. 23 (6), 1789-1792, 2013. Teljes szöveg: https://hdl.handle.net/2437/160558 Folyóirat-mutatók:
Q2 Biochemistry Q2 Clinical Biochemistry Q2 Drug Discovery Q3 Molecular Biology Q3 Molecular Medicine Q2 Organic Chemistry Q1 Pharmaceutical Science | post-print: 192 |
2012 | Nagy, V., Felföldi, N., Kónya, B., Praly, J., Docsa, T., Gergely, P., Chrysina, E., Tiraidis, C., Kosmopoulou, M., Alexacou, K., Konstantakaki, M., Leonidas, D., Zographos, S., Oikonomakos, N., Kozmon, S., Tvaroška, I., Somsák, L.: N-(4-Substituted-benzoyl)-N'-(beta-d-glucopyranosyl)ureas as inhibitors of glycogen phosphorylase: Synthesis and evaluation by kinetic, crystallographic, and molecular modelling methods. Bioorg. Med. Chem. 20 (5), 1801-1816, 2012. Teljes szöveg: https://hdl.handle.net/2437/134810 Folyóirat-mutatók:
Q2 Biochemistry Q1 Clinical Biochemistry Q1 Drug Discovery Q2 Molecular Biology Q2 Molecular Medicine Q1 Organic Chemistry D1 Pharmaceutical Science | post-print: 327 |
2012 | Kónya, B., Docsa, T., Gergely, P., Somsák, L.: Synthesis of heterocyclic N-(beta-d-glucopyranosyl)carboxamides for inhibition of glycogen phosphorylase. Carbohydr. Res. 351 56-63, 2012. Teljes szöveg: https://hdl.handle.net/2437/123684 Folyóirat-mutatók:
Q2 Analytical Chemistry Q3 Biochemistry Q2 Medicine (miscellaneous) Q2 Organic Chemistry | post-print: 145 |
2011 | Docsa, T., Czifrák, K., Hüse, C., Somsák, L., Gergely, P.: Effect of glucopyranosylidene-spiro-thiohydantoin on glycogen metabolism in liver tissues of streptozotocin-induced and obese diabetic rats. Mol. Med. Rep. 4 (3), 477-481, 2011. Teljes szöveg: https://hdl.handle.net/2437/103346 Folyóirat-mutatók:
Q4 Biochemistry Q4 Cancer Research Q4 Genetics Q4 Molecular Biology Q4 Molecular Medicine Q3 Oncology | kiadói változat: 87 |
2011 | Kun, S., Nagy, G., Tóth, M., Czecze, L., Van Nhien, A., Docsa, T., Gergely, P., Charavgi, M., Skourti, P., Chrysina, E., Patonay, T., Somsák, L.: Synthesis of variously coupled conjugates of d-glucose, 1,3,4-oxadiazole, and 1,2,3-triazole for inhibition of glycogen phosphorylase. Carbohydr. Res. 346 (12), 1427-1438, 2011. Teljes szöveg: https://hdl.handle.net/2437/109613 Folyóirat-mutatók:
Q2 Analytical Chemistry Q3 Biochemistry Q2 Medicine (miscellaneous) Q2 Organic Chemistry | post-print: 257 |
2010 | Cheng, K., Liu, J., Sun, H., Bokor, É., Czifrák, K., Kónya, B., Tóth, M., Docsa, T., Gergely, P., Somsák, L.: Tethered derivatives of D-glucose and pentacyclic triterpenes for homo/heterobivalent inhibition of glycogen phosphorylase. New J. Chem. 34 1450-1464, 2010. Teljes szöveg: https://hdl.handle.net/2437/98958 Folyóirat-mutatók:
Q2 Catalysis Q1 Chemistry (miscellaneous) Q1 Materials Chemistry | post-print: 132 |
2009 | Nagy, V., Benltifa, M., Vidal, S., Berzsényi, E., Teilhet, C., Czifrák, K., Batta, G., Docsa, T., Gergely, P., Somsák, L., Praly, J.: Glucose-based spiro-heterocycles as potent inhibitors of glycogen phosphorylase. Bioorg. Med. Chem. 17 (15), 5696-5707, 2009. Teljes szöveg: https://hdl.handle.net/2437/88787 Folyóirat-mutatók:
Q2 Biochemistry Q1 Clinical Biochemistry Q1 Drug Discovery Q3 Molecular Biology Q2 Molecular Medicine Q1 Organic Chemistry Q1 Pharmaceutical Science | post-print: 153 |
2009 | Tóth, M., Kun, S., Bokor, É., Benltifa, M., Tallec, G., Vidal, S., Docsa, T., Gergely, P., Somsák, L., Praly, J.: Synthesis and structure-activity relationships of C-glycosylated oxadiazoles as inhibitors of glycogen phosphorylase. Bioorg. Med. Chem. 17 (13), 4773-4785, 2009. Teljes szöveg: https://hdl.handle.net/2437/87987 Folyóirat-mutatók:
Q2 Biochemistry Q1 Clinical Biochemistry Q1 Drug Discovery Q3 Molecular Biology Q2 Molecular Medicine Q1 Organic Chemistry Q1 Pharmaceutical Science | post-print: 342 |