Publication list
2023
Bokor, É.,
Kecskés, D.,
Gombás, F.,
Fehér, A.,
Kardos, E.,
Dabian, A.,
Vonza, Z.,
Szennyes, E.,
Somsák, L.:
First representatives of C-glycosyl 1,2,4,5-tetrazines: synthesis of 3-beta-d-glucopyranosyl 1,2,4,5-tetrazines and their transformation into 3-beta-d-glucopyranosyl pyridazines.
New Journal of Chemistry 47 (1), 56-74, 2023.
Journal metrics:
Q3 Catalysis
Q2 Chemistry (miscellaneous)
Q2 Materials Chemistry
2021
Sipos, Á.,
Szennyes, E.,
Hajnal, É.,
Kun, S.,
Szabó, E.,
Uray, K.,
Somsák, L.,
Docsa, T.,
Bokor, É.:
Dual-Target Compounds against Type 2 Diabetes Mellitus: proof of Concept for Sodium Dependent Glucose Transporter (SGLT) and Glycogen Phosphorylase (GP) Inhibitors.
Pharmaceuticals. 14 (4), 1-27, 2021.
Journal metrics:
Q1 Drug Discovery
Q2 Molecular Medicine
Q1 Pharmaceutical Science
2020
Kyriakis, E.,
Karra, A.,
Papaioannou, O.,
Solovou, T.,
Skamnaki, V.,
Liggri, P.,
Zographos, S.,
Szennyes, E.,
Bokor, É.,
Kun, S.,
Psarra, A.,
Somsák, L.,
Leonidas, D.:
The architecture of hydrogen and sulfur α-hole interactions explain differences in the inhibitory potency of C-β-d-glucopyranosyl thiazoles, imidazoles and an N-β-d glucopyranosyl tetrazole for human liver glycogen phosphorylase and offer new insights to structure-based design.
Bioorg. Med. Chem. 28 (1), 1-10, 2020.
Journal metrics:
Q3 Biochemistry
Q2 Clinical Biochemistry
Q2 Drug Discovery
Q3 Molecular Biology
Q3 Molecular Medicine
Q2 Organic Chemistry
Q2 Pharmaceutical Science
2019
Barr, D.,
Szennyes, E.,
Bokor, É.,
Al-Oanzi, Z.,
Moffatt, C.,
Kun, S.,
Docsa, T.,
Sipos, Á.,
Davies, M.,
Mathomes, R.,
Snape, T.,
Agius, L.,
Somsák, L.,
Hayes, J.:
Identification of C-[béta]-d-Glucopyranosyl Azole-Type Inhibitors of Glycogen Phosphorylase That Reduce Glycogenolysis in Hepatocytes: in Silico Design, Synthesis, in Vitro Kinetics, and ex Vivo Studies.
ACS Chem. Biol. 14 (7), 1460-1470, 2019.
Journal metrics:
Q1 Biochemistry
D1 Medicine (miscellaneous)
Q1 Molecular Medicine
Szennyes, E.,
Bokor, É.,
Docsa, T.,
Sipos, Á.,
Somsák, L.:
Synthesis of C-β-D-glucopyranosyl derivatives of some fused azoles for the inhibition of glycogen phosphorylase.
Carbohydr. Res. 472 33-41, 2019.
Journal metrics:
Q2 Analytical Chemistry
Q3 Biochemistry
Q2 Medicine (miscellaneous)
Q2 Organic Chemistry
2018
Kun, S.,
Begum, J.,
Kyriakis, E.,
Stamati, E.,
Barkas, T.,
Szennyes, E.,
Bokor, É.,
Szabó, E.,
Stravodimos, G.,
Sipos, Á.,
Docsa, T.,
Gergely, P.,
Moffatt, C.,
Patraskaki, M.,
Kokolaki, M.,
Gkerdi, A.,
Skamnaki, V.,
Leonidas, D.,
Somsák, L.,
Hayes, J.:
A multidisciplinary study of 3-(β-D-glucopyranosyl)-5-substituted-1,2,4-triazole derivatives as glycogen phosphorylase inhibitors: computation, synthesis, crystallography and kinetics reveal new potent inhibitors.
Eur. J. Med. Chem. 147 266-278, 2018.
Journal metrics:
Q1 Drug Discovery
Q1 Medicine (miscellaneous)
Q1 Organic Chemistry
Q1 Pharmacology
Szennyes, E.,
Bokor, É.,
Langer, P.,
Gyémánt, G.,
Docsa, T.,
Sipos, Á.,
Somsák, L.:
The first general synthesis of 2-C-(beta-D-glycopyranosyl)pyrimidines and their evaluation as inhibitors of some glycoenzymes.
New J. Chem. 42 (21), 17439-17446, 2018.
Journal metrics:
Q3 Catalysis
Q2 Chemistry (miscellaneous)
Q1 Materials Chemistry
2017
Szennyes, E.,
Bokor, É.,
Kiss-Szikszai, A.,
Somsák, L.,
Pascal, Y.:
Preparation of 2,6-anhydro-3,4,5,7-tetra-O-benzyl-D-glycero-D-gulo-heptonimidamide.
In: Carbohydrate Chemistry: Proven Synthetic Methods / Christian Vogel, Paul Murphy, CRC Press-Taylor & Francis Group, Boca Raton, 323-332, 2017, (Volume 4 ) ISBN: 9781498726917
2016
Szennyes, E.,
Bokor, É.,
Batta, G.,
Docsa, T.,
Gergely, P.,
Somsák, L.:
Improved preparation of 4(5)-aryl-2-(β-D-glucopyranosyl)-imidazoles, the most efficient glucose analogue inhibitors of glycogen phosphorylase.
RSC Adv. 6 (97), 94787-94794, 2016.
Journal metrics:
Q1 Chemical Engineering (miscellaneous)
Q1 Chemistry (miscellaneous)
2015
Bokor, É.,
Szennyes, E.,
Csupász, T.,
Tóth, N.,
Docsa, T.,
Gergely, P.,
Somsák, L.:
C-(2-Deoxy-D-arabino-hex-1-enopyranosyl)-oxadiazoles: synthesis of possible isomers and their evaluation as glycogen phosphorylase inhibitors.
Carbohydr. Res. 412 71-79, 2015.
Journal metrics:
Q2 Analytical Chemistry
Q3 Biochemistry
Q2 Medicine (miscellaneous)
Q2 Organic Chemistry
updated: 2024-11-09, 01:44